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Kinetics of Enzyme Action - Basic Principles for Drug Hunters |
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| Course Code: KNTX |
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| This course covers the essentials of enzyme kinetic analysis emphasizing concepts of importance in drug discovery. It provides an introduction to enzymology, assay methods, and free-energy diagrams; and also covers simple reversible inhibition and time-dependent inhibition; transition state rate theory and TS analog inhibitors; kinetics and inhibition of two substrate enzymatic reactions; screening for inhibitors of enzymatic reactions; and, probes of mechanism. |
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Dates - TBA |
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Check-in opens at 7:30 a.m. on the first day of the course.
Course runs from 8:30 a.m. to 5:00 p.m. each day. |
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Event Location: |
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TBA |
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Early Registration: |
$1,295 |
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Advanced Registration: |
$1,395 |
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Standard Registration: |
$1,495 |
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The course fee includes a course binder and a continental breakfast each day.
Five for Four! Register five people for one course, one person for five courses, or any combination in between and your fifth registration is free. Note: This discount is only available if you register by fax or mail and mention this discount. May not be combined with any other offer. |
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- Enzymology, Assay Methods, and Free-Energy Diagrams
- Concepts of Simple Reversible Inhibition
- Time-Dependent Inhibition
- Transition State Rate Theory and TS Analog Inhibitors
- Kinetics of Two Substrate Enzymatic Reactions
- Inhibition of Two-Substrate Enzymatic Reactions
- Screening for Inhibitors of Enzymatic Reactions
- Probes of Mechanism
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| Ross Stein is an Associate Professor in the Department of Neurology at Harvard Medical School and Director of the Laboratory for Drug Discovery in Neurodegeneration of the Harvard Center for Neurodegeneration and Repair. He teaches Kinetics of Enzyme Action - Basic Principles for Drug Hunters. |
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